Their use for the 4-pyridinone compounds and cancer

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专利权人:

ブリストル－マイヤーズ;スクイブ;ブリストル-マイヤーズ スクイブ カンパニー;カンパニー

发明人:

ロバート・シー・リビングストン,ウィリアム・ピー・ギャラガー

申请号：

JP2010544406

公开号：

JP5693239B2

申请日:

2009.01.22

申请国别(地区):

JP

年份:

2015

代理人:

摘要：

Disclosed herein is a process for preparing a compound of Formula (I), comprising the steps of: (a) reacting an aniline compound of Formula (II) and an carboxylic acid compound of Formula (III) or an activated carboxylic acid compound thereof, to provide a compound of Formula (IV)； and (b) converting said protected amine group attached to said compound of Formula (IV) to an amine group to provide said compound of Formula (I)； wherein PAm is a protected amine group. Processes to prepare the compounds of Formulae (II), (III), and (IV) are also disclosed.

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