您的位置: 首页 > 农业专利 > 详情页

PYRROLO-DIAZEPINES ET PYRAZOLO-DIAZEPINES SUBSTITUEES EN POSITION 4
专利权人:
BAYER PHARMA AKTIENGESELLSCHAFT
发明人:
SCHMEES, NORBERT,BUCHMANN, BERND,HAENDLER, BERNARD,NEUHAUS, ROLAND,LEJEUNE, PASCALE,KRUGER, MARTIN,FERNANDEZ-MONTALVAN, AMAURY ERNESTO,KUNZER, HERMANN (DECEASED),REHWINKEL, HARTMUT
申请号:
CA2901805
公开号:
CA2901805A1
申请日:
2014.02.18
申请国别(地区):
CA
年份:
2014
代理人:
摘要:
BET-protein-inhibiting, in particular BRD2-, BRD3- and BRD4-inhibiting 4-substituted pyrrolo- and pyrazolo-diazepines, of general formula I in which X, Y, n, m, p, R1, R2, R3, R4 and R5 have the meanings indicated in the description, pharmaceutical agents containing the compounds according to the invention and the prophylactic and therapeutic use thereof for treating hyperproliferative diseases, in particular tumor diseases, are described. Furthermore, the use of the compounds according to the invention as BET-protein inhibitors in benign hyperplasias, in atherosclerotic diseases, in sepsis, in autoimmune diseases, in vascular diseases, in viral infections, in neurodegenerative diseases, in inflammatory diseases, in atherosclerotic diseases and for controlling fertility in males is described.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充