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FUSED SUBSTITUTE AMINOPYRROLIDINE DERIVATIVE
专利权人:
DAIICHI SANKYO COMPANY; LIMITED
发明人:
HISASHI TAKAHASHI,RIE MIYAUCHI,MASATOSHI NAGAMOCHI,SATOSHI KOMORIYA,TAKAHIRO KITAMURA,TAKASHI ODAGIRI,HIROAKI INAGAKI,TOSHIFUMI TSUDA,KIYOSHI NAKAYAMA,MAKOTO TAKEMURA,KENICHI YOSHIDA
申请号:
MYPI 20092809
公开号:
MY162052A
申请日:
2007.12.28
申请国别(地区):
MY
年份:
2017
代理人:
摘要:
A QUINOLONE SYNTHETIC ANTIBACTERIAL AGENT HAVING EXCELLENT PROPERTIES AS A MEDICINE IS PROVIDED, WHICH HAS STRONG ANTIBACTERIAL ACTIVITY NOT ONLY TO GRAM-NEGATIVE BACTERIA BUT ALSO TO GRAM-POSITIVE COCCI THAT HAVE LOW SENSITIVITY TO QUINOLONE ANTIBACTERIAL AGENTS, AND WHICH EXHIBITS HIGH SAFETY AND EXCELLENT PHARMACOKINETICS. A COMPOUND REPRESENTED BY THE FORMULA (I) OR A SALT THEREOF, OR A HYDRATE THEREOF. SPECIFICALLY, A QUINCLONE DERIVATIVE OF THE FORMULA (I) WHEREIN SUBSTITUENTS R6 AND R7 TAKEN TOGETHER WITH THE CARBON ATOMS TO WHICH THEY ARE BONDED FORM A CYCLIC STRUCTURE WHICH MAY CONTAIN AN OXYGEN ATOM AS A RING CONSTITUENT ATOM, THE CYCLIC STRUCTURE FORMING A 5- 4, 5-5, OR 5-6 FUSED BICYCLIC PYRROLIDINYL SUBSTITUENT, THE SUBSTITUENT BEING BONDED TO A QUINOLONE MOTHER SKELETON Q CONTAINING A PYRIDOBENZOXAZINE STRUCTURE:
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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