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compound, pharmaceutical composition, use of a compound, and method
专利权人:
MERCK SHARP & DOHME CORP.
发明人:
Amjad Ali,Andrew Stamford,Christopher Boyce,Dong Xiao,Edward Metzger,Gioconda V. Gallo,Heping Wu,Jae-Hun Kim,Junying Zheng,Michael Man-Chu Lo,Nicolas Zorn,Paul Tempest,Pauline Ting,Qiaolin Deng,Rongze
申请号:
BR112015015468
公开号:
BR112015015468A2
申请日:
2013.12.20
申请国别(地区):
BR
年份:
2017
代理人:
摘要:
1/1 summary "compound, pharmaceutical composition, use of a compound, and method" are described compounds of the formula g1 (structurally represented): where "rg3", "rd1" â € œrd4â €, â € œnâ €, â € œmâ €, â € œpâ €, â € œwâ €, â € œxâ €, â € œyâ € and â € œsaneâ € as defined herein, which compounds are α 2α receptor antagonists. Also described herein are the uses of the compounds described herein as α2α receptor antagonists in the potential treatment or prevention of neurological disorders and disorders in which α2α receptors are involved. Also disclosed herein are pharmaceutical compositions comprising these compounds and uses of these pharmaceutical compositions.1 / 1 resumo “composto, composiã‡ãƒo farmacãšutica, uso de um composto, e, mã‰todoâ€� sã£o descritos compostos da fã³rmula g1 (estruturalmente representados): onde “rg3â€�, “rd1â€� a “rd4â€�, “nâ€�, “mâ€�, “pâ€�, “wâ€�, “xâ€�, “yâ€� e “zâ€� sã£o aqui definidos, compostos estes que sã£o antagonistas do receptor de a2a. tambã©m sã£o aqui descritos os usos dos compostos aqui descritos como antagonistas do receptor de a2a no tratamento ou prevenã§ã£o potenciais de distãºrbios e doenã§as neurolã³gicas em que os receptores de a2a estã£o envolvidos. tambã©m sã£o aqui descritas composiã§ãµes farmacãªuticas compreendendo estes compostos e usos destas composiã§ãµes farmacãªuticas.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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