HANAGAN, MARY ANN,OBERHOLZER, MATTHEW RICHARD,PASTERIS, ROBERT JAMES,SHAPIRO, RAFAEL
申请号：
CA2757055
公开号：
CA2757055C
申请日:
2010.04.19
申请国别(地区):
CA
年份:
2017
代理人:
摘要：
Disclosed are solid forms of 1-[4-[4-[5-(2,6-difluorophenyl)-4,5-dihydro-3-isoxazolyl]-2-thiazolyl]-1-piperidinyl]-2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethanon e(Compound 1). Methods for the preparation of solidforms of Compound 1 and for the conversion of one solid form of Compound 1into another are disclosed. Disclosed are fungicidalcompositions comprising a fungicidally effective amount of a solid form ofCompound 1 and at least one additional componentselected from the group consisting of surfactants, solid diluents and liquidcarriers. Compositions comprising a mixture of asolid form of Compound 1 and at least one other fungicide or insecticide arealso disclosed. Also disclosed are methods for controllingplant diseases caused by fungal plant pathogens comprising applying to a plantor portion thereof, or to a plant seed, afungicidally effective amount of a solid form of Compound 1.
