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Triazole compounds and preparation and use procedures
- 专利权人:
- Inc.;Melinta Therapeutics
- 发明人:
- BHATTACHARJEE, Ashoke,KANYO, Zoltan F.,SHERER, Edward C.
- 申请号：
- ES06802533
- 公开号：
- ES2638427T3
- 申请日:
- 2006.08.24
- 申请国别(地区):
- ES
- 年份:
- 2017
- 代理人:
- 摘要：
- A compound having the structure: ** Formula ** or a salt, ester or N-oxide thereof, in which A is selected from: (a) a C1-6 alkyl group, (b) a C2 alkenyl group -6, (c) a C2-6 alkynyl group, (d) a C3-12 saturated, unsaturated or aromatic carbocycle, (e) a 3-12 membered saturated, unsaturated or aromatic heterocycle containing one or more nitrogen atoms , oxygen or sulfur, (f) H, (g) -OH, (h) -SH, (i) F, (j) Cl, (k) Br, (l) I, (m) -CF3, (n ) -CN, (o) -N3, (p) NO2, (q) -NR6 (CR6R6) tR9, (r) -OR9, (s) -S (CR6R6) tR9, (t) -C (O) ( CR6R6) tR9, (u) -OC (O) (CR6R6) tR9, (v) - OC (O) O (CR6R6) tR9, (w) -SC (O) (CR6R6) tR9, (x) -C ( O) O (CR6R6) tR9, (y) - NR6C (O) (CR6R6) tR9, (z) -C (O) NR6 (CR6R6) tR9, (aa) -C (>； = NR6) (CR6R6) tR9, (bb) -C (>； = NNR6R6) (CR6R6) tR9, (cc) - C [>； = NNR6C (O) R6] (CR6R6) tR9, (dd) -NR6C (O) O (CR6R6) tR9, (ee ) -OC (O) NR6 (CR6R6) tR9, (ff) - NR6C (O) NR6 (CR6R6) tR9, (gg) -NR6S (O) p (CR6R6) tR9, (hh) -S (O) pNR6 ( CR6R6) tR9, (ii) -NR6R6, (jj) -SR6, (kk) -S (O) R6, (ll) NR6C (O) R6, (mm) -Si (R13) 3 and ( nn) -C (>； = O) H, in which (a) - (e) are optionally substituted by one or more R14 groups； T is ** Formula ** in which: M is selected from: (a) -C (O) -, (b) -CH (-OR114) -, (c) -NR114-CH2-, (d) -CH2-NR114-, (e) - CH (NR114R114) -, (f) -C (>； = NNR114R114) -, (g) -NR114-C (O) -, (h) -C (O) NR114- , (i) - C (>； = NR114) -, (j) -CR115R115- and (k) -C (>； = NOR127) -； R100 is selected from (a) H, (b) F, (c) Cl, (d) Br, (e) -SR114 and (f) C1-6 alkyl, in which (f) is optionally substituted by one or more R115 groups； R101 is selected from: (a) H, (b) Cl, (c) F, (d) Br, (e) I, (f) -NR114R114, (g) -NR114C (O) R114, (h) -OR114, (i) -OC (O) R114, (j) - OC (O) OR114, (k) -OC (O) NR114R114, (l) -O-C1-6 alkyl, (m) -OC ( O) -C 1-6 alkyl, (n) -OC (O) O-C 1-6 alkyl, (o) -OC (O) NR114-C 1-6 alkyl, (p) C 1-6 alkyl, (q) alkenyl C1-6 and (r) C1-6 alkynyl, wherein any of (l) - (r) is optionally substituted by one or more R115 groups； R102 is
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- 中国工程科技知识中心
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