您的位置: 首页 > 农业专利 > 详情页

Heteroaryl-carboxylic acid (sulfamoylalkyl) amide derivatives as factor Xa inhibitors
专利权人:
サノフイ
发明人:
ミヒャエル・ヴァーグナー,マティーアス・ウーアマン,フォルクマール・ヴェーナー,マルティン・ロレンツ,アルミン・バウアー,マルク・ナザレ,ハンス・マター
申请号:
JP2008511587
公开号:
JP5027802B2
申请日:
2006.05.06
申请国别(地区):
JP
年份:
2012
代理人:
摘要:
The present invention relates to compounds of the formula I, in which R1; R2; R3; V; G1 and G2 have the meanings indicated in the claims. The compounds of the formula I are valuable pharmacologically active compounds. They exhibit a strong antithrombotic effect and are suitable, for example, for the therapy and prophylaxis of cardiovascular disorders like thromboembolic diseases or restenoses. They are reversible inhibitors of the blood clotting enzymes factor Xa, and can in general be applied in conditions in which an undesired activity of factor Xa is present or for the cure or prevention of which an inhibition of factor Xa is intended. The invention furthermore relates to processes for the preparation of compounds of the formula I, their use, in particular as active ingredients in pharmaceuticals, and pharmaceutical preparations comprising them.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充