ENTWISTLE, DAVID, ANDREW,MARSHALL, PETER, WALLANCE,TAYLOR, STEFAN, COLIN, JOHN
申请号:
HK08106870.4
公开号:
HK1116485B
申请日:
2008.06.20
申请国别(地区):
HK
年份:
2012
代理人:
摘要:
The invention comprises (1) anhydrous crystalline forms of N-[1-(2-ethoxyethyl)-5-(N-ethyl-N-methylamino)-7-(4-methylpyridin-2-yl-amino)-1H-pyrazolo[4,3-d]pyrimidine-3-carbonyl]methanesulfonamide, (2) pharmaceutical compositions comprising at least one such form, (3) methods for the treatment of a phosphodiesterase-5-mediated condition using at least one such form, and (4) methods for preparing such forms. The compound N-[1-(2-ethoxyethyl)-5-(N-ethyl-N-methylamino)-7-(4-methylpyridin-2-yl-amino)-1H-pyrazolo[4,3-d]pyrimidine-3-carbonyl]methanesulfonamide has the following structure (I).