MOUND, William Roderick,SCUTT, James Nicholas,SLATER, Mark,WILLETTS, Nigel James
申请号：
ES13811960
公开号：
ES2665568T3
申请日:
2013.12.19
申请国别(地区):
ES
年份:
2018
代理人:
摘要：
A compound of formula (I): ** (See formula) **, wherein: X is methyl or chlorine； R1 is methyl or chlorine； R2 is hydrogen, methyl, ethyl, n-propyl, cyclopropyl, vinyl, ethynyl, fluorine, chlorine, bromine, C1-C3 alkoxy, fluoroalkoxyC1-C2, C1-C2-alkoxyC1-C3- or fluoroalkoxyC1-alkoxyC1-C3-； and R3, R4, R5 and R6, independently of one another, are hydrogen, C1-C5 alkyl, C2-C4 alkenyl, C2-C4 alkynyl, C1-C2 fluoroalkyl, C1-C3 alkoxyC1-C3-alkyl, C1-C3-C3-C3-C1-C3-alkyl C1-1C3 alkyl sulfonylalkyl C1-C3 alkyl； C3-C4 cycloalkyl； or an unsubstituted monocyclic 4-, 5- or 6-membered heterocyclyl having a ring heteroatom independently selected from oxygen, sulfur and nitrogen and attached to a ring carbon atom within the heterocyclyl； provided that no more than one of R3, R4, R5 and R6 is alkenyl, alkynyl, alkoxyalkyl, alkylthioalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl, cycloalkyl or heterocyclyl； or R3 and R4 taken together are - (CH2) n1- or - (CH2) n2-X1- (CH2) n3- and R5 and R6 are as defined herein, or R5 and R6 taken together are - (CH2 ) n1- or - (CH2) n2-X1- (CH2) n3- and R3 and R4 are as defined herein； wherein X1 is O, S, S (O), S (O) 2, NH, N (C1-C2 alkyl), N (C1-C2 alkoxy), C (H) (C1-C2 alkyl), C (C1-C2 alkyl ) 2 or C (H) (C1-C2 alkoxy)； n1 is 2, 3, 4 or 5； and n2 and n3 are independently 1, 2 or 3 as long as n2 + n3 is 2, 3 or 4； or R4 and R5 taken together are - (CH2) n4- or - (CH2) n5-C (R7a) (R7b) - (CH2) n6- or -C (R7c)>； = C (R7d) -； wherein R7a is C1-C2 alkyl or C1-C2 alkoxy； and R7b is hydrogen or C1-C2 alkyl provided that R7b is hydrogen when R7a is C1-C2 alkoxy； n4 is 1, 2 or 3； and n5 and n6 are independently 0, 1 or 2 provided that n5 + n6 is 0, 1 or 2； and R7c and R7d are independently hydrogen or C1-C2 alkyl； and Y is O, S, S (O), S (O) 2, N (C1-C2 alkyl), N (C1-C2 alkoxy), C (O), CR8R9 or -CR10R11CR12R13-； and R8 and R9 are independently hydrogen, C1-C6alkyl, C2-C4 alkenyl, C4-alquiniloC2, fluoroalquiloC1-C2-C3 alcoxiC1-C3alquiloC1, alquilC1- C3
