ARORA, Paramjit S.,LAO, Brooke Bullock,HENCHEY, Laura K.,TRAASETH, Nathaniel J.,THOMSON, Paul,KUSHAL, Swati,OLENYUK, Bogdan Z.
申请号:
EP14843057
公开号:
EP3041492A4
申请日:
2014.09.03
申请国别(地区):
EP
年份:
2017
代理人:
摘要:
The present invention relates to peptidomimetics that mimic helix &alphaB of the C-terminal transactivation domain of HIF-1&alpha. Methods of using the peptidomimetics to, e.g., inhibit the HIF-1&alpha-p300/CBP interaction, are also disclosed.