DE KOCK, HERMAN,JONCKERS, TIM HUGO MARIA,BOONANTS, PAUL JOZEF GABRIEL MARIA,LAST, STEFAAN JULIEN,DIERYNCK, INGE,BAUMEISTER, JUDITH EVA,VAN 'T KLOOSTER, GERBEN ALBERT ELEUTHERIUS,DE KOCK HERMAN,JONCKERS TIM HUGO MARIA,BOONANTS PAUL JOZEF GABRIEL MARIA,LAST STEFAAN JULIEN,DIERYNCK INGE
申请号:
PL07765554
公开号:
PL2035432T3
申请日:
2007.06.22
申请国别(地区):
PL
年份:
2012
代理人:
摘要:
The present invention relates to 2-(substituted-amino)-benzothiazole sulfonamide compounds and derivatives, their use as protease inhibitors, in particular as broad-spectrum HIV protease inhibitors, processes for their preparation as well as pharmaceutical compositions and diagnostic kits comprising them. The present invention also concerns combinations of the present 2-(substituted-amino)-benzothiazole sulfonamide compounds and derivatives with another anti-retroviral agent. It further relates to their use in assays as reference compounds or as reagents.