DE KOCK, HERMAN AUGUSTINUS,JONCKERS, TIM HUGO MARIA,BOONANTS, PAUL JOZEF GABRIEL MARIA,LAST, STEFAAN JULIEN,DIERYNCK, INGE,BAUMEISTER, JUDITH EVA,VAN T KLOOSTER, GERBEN ALBERT ELEUTHERIUS
申请号：
MYPI 20085209
公开号：
MY146805A
申请日:
2007.06.22
申请国别(地区):
MY
年份:
2012
代理人:
摘要：
THE PRESENT INVENTION RELATES TO 2-(SUBSTITUTED-AMINO)-BENZOTHIAZOLE SULFONAMIDE COMPOUNDS AND DERIVATIVES, THEIR USE AS PROTEASE INHIBITORS, IN PARTICULAR AS BROADSPECTRUM HIV PROTEASE INHIBITORS, PROCESSES FOR THEIR PREPARATION AS WELL AS PHARMACEUTICAL COMPOSITIONS AND DIAGNOSTIC KITS COMPRISING THEM. THE PRESENT INVENTION ALSO CONCERNS COMBINATIONS OF THE PRESENT 2-(SUBSTITUTED-AININO)-BENZOTHIAZOLE SULFONAMIDE COMPOUNDS AND DERIVATIVES WITH ANOTHER ANTI-RETROVIRAL AGENT. IT FURTHER RELATES TO THEIR USE IN ASSAYS AS REFERENCE COMPOUNDS OR AS REAGENTS.
