DE KOCK HERMAN,JONCKERS TIM HUGO MARIA,BOONANTS PAUL JOZEF GABRIEL MARIA,LAST STEFAAN JULIEN,DIERYNCK INGE,BAUMEISTER JUDITH EVA,VAN T KLOOSTER GERBEN ALBERT ELEUTHERIUS
申请号:
SI200730904
公开号:
SI2035432T1
申请日:
2007.06.22
申请国别(地区):
SI
年份:
2012
代理人:
摘要:
The present invention relates to 2-(substituted-amino)-benzothiazole sulfonamide compounds and derivatives, their use as protease inhibitors, in particular as broad-spectrum HIV protease inhibitors, processes for their preparation as well as pharmaceutical compositions and diagnostic kits comprising them. The present invention also concerns combinations of the present 2-(substituted-amino)-benzothiazole sulfonamide compounds and derivatives with another anti-retroviral agent. It further relates to their use in assays as reference compounds or as reagents.