GONZALEZ-BOBES, FRANCISCO,BULTMAN, MICHAEL S.,COHEN, BENJAMIN,HICKEY, MATTHEW R.
申请号:
CA2971096
公开号:
CA2971096A1
申请日:
2015.12.17
申请国别(地区):
CA
年份:
2016
代理人:
摘要:
A process for preparing halogenated azaindole compounds makes use of a brominating agent PyBroP, together with a dehydrating agent BSA to enhance the selectivity and improve the yield of the final product which is a piperazine prodrug useful as an antiviral.