Gonzalez-Bobes, Francisco,Bultman, Michael S.,Cohen, Benjamin,Hickey, Matthew R.
申请号:
AU2015364535
公开号:
AU2015364535A1
申请日:
2015.12.17
申请国别(地区):
AU
年份:
2017
代理人:
摘要:
A process for preparing halogenated azaindole compounds makes use of a brominating agent PyBroP, together with a dehydrating agent BSA to enhance the selectivity and improve the yield of the final product which is a piperazine prodrug useful as an antiviral.