COOYMANS, Ludwig Paul,DEMIN, Samuël Dominique,HU, Lili,JONCKERS, Tim Hugo Maria,RABOISSON, Pierre Jean-Marie Bernard,TAHRI, Abdellah,VENDEVILLE, Sandrine Marie Helene
申请号：
ES11794793
公开号：
ES2572258T3
申请日:
2011.12.16
申请国别(地区):
ES
年份:
2016
代理人:
摘要：
A compound of formula (I), a N -oxide, addition salt, quaternary amine, metal complex or stereochemically isomeric form thereof ** ** Formula where each X is independently C or N R1 is selected from the group of H, halogen, C1-C6 alkoxy, CF3 and OCF3 R2 is selected from the group consisting of H, halogen, C1-C6 alkyl, C3-C7 cycloalkyl, C1-C6 alkoxy and CO (R7) R3 is - (CR8R9) n-R10 R4 is selected from the group consisting of H, C1-C10 alkyl, C3-C7 cycloalkyl, C2-C10 alkenyl, SO2-R8, CH2CF3, SO2CH3 or a saturated ring of 4 to 6 members containing one oxygen atom R5 is present when X is C and is selected from the group consisting of H, C1-C6 alkyl, C3-C7 cycloalkyl, C1-C6 alkyl, CO (R7), CF3 and halogen R5 is absent when X is N R7 is I selected from the group consisting of OH, O (C1-C6) alkyl, NH2, NHSO2N (C1-C6) 2, NHSO2NHCH3, NHSO2 (C1-C6), NHSO2 (C3-C7) and N (alkyl C1-C6) 2, NR8R9, NR9R10 n is an integer from 2 to 6 R8 and R9 are each independently selected from H, C1-C10 alkyl, C3-C7 cycloalkyl or R8 and R9 taken together form an aliphatic ring of 4 to 6 members optionally containing one or more heteroatoms selected from N, S, O R10 is selected from the group consisting of H, C1-C6, OH, CN, F, CF2H, CF3, C (> = NOH) NH2, CONR8R9, COOR8, CONR8SO2R9, CON (R8) SO2N (R8R9) NR8R9, NR8COOR9, OCOR8, NR8SO2R9, SO2NR8R9, SO2R8 or a saturated ring of 4 to 6 members containing one oxygen atom.Un compuesto de fórmula (I), un N-óxido, una sal por adición, una amina cuaternaria, un complejo metálico o una forma estereoquímicamente isómera del mismo **Fórmula** en donde cada X es independientemente C o N R1 se selecciona del grupo de H, halógeno, alcoxi C1-C6, CF3 y OCF3 R2 se selecciona del grupo que consiste en H, halógeno, alquilo C1-C6, cicloalquilo C3-C7, alcoxi C1-C6 y CO(R7) R3 es -(CR8R9)n-R10 R4 se selecciona del grupo que consiste en H, alquilo C1-C10, cicloalquilo C3-C7, alquenilo C2-C10, SO2-R8, CH2CF3, SO2CH3 o un anillo saturado de 4 a 6 miembros que contiene un
