COOYMANS, Ludwig Paul,DEMIN, Samuël Dominique,HU, Lili,JONCKERS, Tim Hugo Maria,RABOISSON, Pierre Jean-Marie Bernard,TAHRI, Abdellah,VENDEVILLE, Sandrine Marie Helene
申请号：
ES11802054
公开号：
ES2576180T3
申请日:
2011.12.16
申请国别(地区):
ES
年份:
2016
代理人:
摘要：
A compound represented by formula I, an N-oxide, salt by addition, quaternary amine, metal complex or a stereochemically isomeric form thereof: ** Formula ** wherein each of the X, independently, is C or N； R1 is H； R2 is selected from the group consisting of Br and Cl； R3 is - (CR6R7) n-R8； R4 is selected from the group consisting of C3-C7 cycloalkyl, C2-C10 alkenyl, CH2CF3 and -SO2CH3； R5 is present in cases where X is C, where each of the R5 is each independently selected from the group consisting of H, C1-C6 alkyl, C1-C6 alkoxy, halogen and CN； R5 is absent in cases where X is N； R6 and R7 are each independently selected from H and C1-C10 alkyl, cycloalkyl, C3-C7； or R6 and R7, taken together, form a 5- to 6-membered aliphatic or aromatic ring that optionally contains one or more heteroatoms selected from the group N, S, O； R8 is selected from the group consisting of H, OH, CF3, CHF2, F, Cl, SO2CH3, SO2cycloalkyl C3-C7, NR6SO2R6, SO2NR6R7, NR6SO2cycloalkyl C3-C7, CN, NR6R7, COOH, COOR6, CONR6R7- OCOalkyl C6, CONR6SO2R7, CONH-R6-SO2R7, CONH-R6-SO2NR6R7CONR6SO2NR6R7, phthalimido or an aliphatic or aromatic ring of 5 to 6 members, optionally containing one or more heteroatoms selected from the group N, S, O； n is an integer that has a value from 1 to 6.Un compuesto representado por la fórmula I, un N-óxido, sal por adición, amina cuaternaria, complejo metálico o una forma estereoquímicamente isomérica del mismo:**Fórmula** en donde cada uno de los X, independientemente, es C o N； R1 es H； R2 se selecciona del grupo que consiste en Br y Cl； R3 es -(CR6R7)n-R8； R4 se selecciona del grupo que consiste en cicloalquilo C3-C7, alquenilo C2-C10, CH2CF3 y -SO2CH3； R5 está presente en los casos en los que X es C, en que cada uno de los R5 se selecciona, cada uno independientemente, del grupo que consiste en H, alquilo C1-C6, alcoxi C1-C6, halógeno y CN； R5 está ausente en los casos en los que X es N； R6 y R7 se seleccionan, cada uno independientemente, de H y alquilo C1-C10
