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glycosidase inhibitors and their uses
- 专利权人:
- ALECTOS THERAPEUTICS INC.;MERCK SHARP & DOHME CORP.
- 发明人:
- David J. Vocacllo,Ernest J. Mceachern,Harold G. Selnick,Qun Dang,Ramesh Kaul,Yuanxi Zhou
- 申请号:
- BR112015009638
- 公开号:
- BR112015009638A2
- 申请日:
- 2013.10.30
- 申请国别(地区):
- BR
- 年份:
- 2017
- 代理人:
- 摘要:
- Summary of the Patent for "Glycosidase Inhibitors and Uses of Them" The invention provides compounds with increased permeability to selectively inhibit glycosidases, prodrugs of the compounds, and compositions. Pharmaceutical compositions including the compounds or prodrugs of the compounds The invention also provides methods of treating diseases and disorders related to o-glycase deficiency or overexpression, accumulation O-glcnac deficiency or impairment.resumo da patente de invenã§ã£o para: “inibidores de glicosidase e usos dos mesmos". a invenã§ã£o proporciona compostos com permeabilidade aumentada para inibir seletivamente as glicosidases, prã³-fã¡rmacos dos compostos, e composiã§ãµes farmacãªuticas incluindo os compostos ou prã³-fã¡rmacos dos compostos. a invenã§ã£o tambã©m proporciona mã©todos de tratamento de doenã§as e distãºrbios relacionados com a deficiãªncia ou a superexpressã£o de o-glcnacase, acumulaã§ã£o ou deficiãªncia de o-glcnac.
- 来源网站:
- 中国工程科技知识中心
- 来源网址:
- http://www.ckcest.cn/home/