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AMINO QUINAZOLINES DERIVATIVES WITH BLOOD PLATELET REDUCING PROPERTIES
专利权人:
发明人:
FRANKLIN, RICHARD,GOLDING, BERNARD
申请号:
MYPI 20092152
公开号:
MY149620A
申请日:
2007.11.19
申请国别(地区):
MY
年份:
2013
代理人:
摘要:
THIS INVENTION RELATES TO THE DISCOVERY OF PRODRUGS OF 3-OR 5-SUBSTITUTED ANALOGUES OF THE SELECTIVE PLATELET LOWERING AGENT ANAGRELIDE WHICH HAVE REDUCED POTENTIAL FOR CARDIOVASCULAR SIDE-EFFECTS AND WHICH SHOULD THEREFORE LEAD TO IMPROVED PATIENT COMPLIANCE AND SAFETY IN THE TREATMENT OF MYELOPROLIFERATIVE DISEASES. MORE SPECIFICALLY, THE PRESENT INVENTION RELATES TO PRODRUGS OF CERTAIN IMIDAZOQUINAZOLINE DERIVATIVES WHICH HAVE UTILITY AS PLATELET LOWERING AGENTS IN HUMANS. THE COMPOUNDS OF THE PRESENT INVENTION FUNCTION BY INHIBITING THE FORMATION OF BLOOD PLATELET.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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