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PHARMACEUTICAL FORMULATION 514
专利权人:
发明人:
BECHTOLD, MICHAEL, KARL,PACKHAEUSER, CLAUDIA, BETTINA,CAHILL, JULIE, KAY,FASTNACHT, KATJA, MAREN,LIEPOLD, BERND, HARALD,LENNON, KIERAN, JAMES,STEITZ, Benedikt
申请号:
MYPI 2011001567
公开号:
MY160340A
申请日:
2009.10.05
申请国别(地区):
MY
年份:
2017
代理人:
摘要:
THE PRESENT INVENTION RELATES TO A PHARMACEUTICAL FORMULATION COMPRISING THE DRUG 4-[3-(4- CYCLOPROPANECARBONYL-PIPERAZINE- 1 -CARBONYL)-4-FLUORO-BENZYL] -2H-PHTHALAZI N-1 -ONE IN A SOLID DISPERSION WITH A MATRIX POLYMER THAT EXHIBITS LOW HYGROSCOPICITY AND HIGH SOFTENING TEMPERATURE, SUCH AS COPOVIDONE. THE INVENTION ALSO RELATES TO A DAILY PHARMACEUTICAL DOSE OF THE DRUG PROVIDED BY SUCH A FORMULATION. IN ADDITION, THE INVENTION RELATES TO THE USE OF A MATRIX POLYMER THAT EXHIBITS LOW HYGROSCOPICITY AND HIGH SOFTENING TEMPERATURE IN SOLID DISPERSION WITH 4-[3-(4-CYCLOPROPANECARBORIYL-PIPERAZINE- 1 -CARBONYL)-4-FLUORO-BENZYL]-2H- PHTHALAZIN-1 -ONE FOR INCREASING THE BIOAVAILABILITY OF THE DRUG.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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