CASIMIRO-GARCIA, AGUSTIN,COE, JOTHAM WADSWORTH,LEFKER, BRUCE ALLEN,NARAYANAN, ARJUN VENKAT,PAPAIOANNOU, NIKOLAOS
申请号:
CA2933026
公开号:
CA2933026A1
申请日:
2016.06.15
申请国别(地区):
CA
年份:
2016
代理人:
摘要:
Disclosed are novel pyridine pyrazinones or pharmaceutically acceptable saltsthereof.Pharmaceutical compositions and the use of the compounds as inhibitors ofBRD4, a member ofthe BET family bromodomain, are also disclosed. Methods for preparing thesecompounds arefurther described.