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new compounds
- 专利权人:
- Chiesi Farmaceutici S.p.A.
- 发明人:
- ALCARAZ, Lilian,HEALD, Robert Andrew,SUTTON, Jonathan Mark,ARMANI, Elisabetta,CAPALDI, Carmelida
- 申请号:
- ES14731580
- 公开号:
- ES2670018T3
- 申请日:
- 2014.06.12
- 申请国别(地区):
- ES
- 年份:
- 2018
- 代理人:
- 摘要:
- A compound selected from the group consisting of 1- (2- {5-cyano-2 - [(R) -6-methoxycarbonyl-7-methyl-3-oxo-8- (3-trifluoromethylphenyl) -2,3 bromide , 5,8-tetrahydro- [1,2,4] triazolo [4,3a] pyrimidin-5-yl] -phenyl} -ethyl) -4-methoxy-pyridinium; 1- (2- {5-Cyano-2 - [(R) -6-methoxycarbonyl-7-methyl-3-oxo-8- (3-trifluoromethylphenyl) -2,3,5,8-tetrahydro- [ 1,2,4] triazolo [4,3-a] pyrimidin-5-yl] -phenyl} -ethyl) -3-hydroxy-pyridinium; 1- (2- {5-Cyano-2 - [(R) -6-methoxycarbonyl-7-methyl-3-oxo-8- (3-trifluoromethylphenyl) -2,3,5,8-tetrahydro- [ 1,2,4] triazolo [4,3-a] pyrimidin-5-yl] -phenyl} -ethyl) -2-methylpyridinium; 1- (2- {5-Cyano-2 - [(R) -6-methoxycarbonyl-7-methyl-3-oxo-8- (3-trifluoromethylphenyl) -2,3,5,8-tetrahydro- [ 1,2,4] triazolo [4,3-a] pyrimidin-5-yl] -phenyl} -ethyl) -4-hydroxymethyl-pyridinium; 1- (2- {5-Cyano-2 - [(R) -6-methoxycarbonyl-7-methyl-3-oxo-8- (3-trifluoromethylphenyl) -2,3,5,8-tetrahydro- [ 1,2,4] triazolo [4,3-a] pyrimidin-5-yl] -phenyl} -ethyl) -4-isopropyl-pyridinium; 1- (2- {5-Cyano-2 - [(R) -6-methoxycarbonyl-7-methyl-3-oxo-8- (3-trifluoromethylphenyl) -2,3,5,8-tetrahydro- [ 1,2,4] triazolo [4,3-a] pyrimidin-5-yl] -phenyl} -ethyl) -5-hydroxy-2-methyl-pyridinium; 1- (2- {5-Cyano-2 - [(R) -6-methoxycarbonyl-7-methyl-3-oxo-8- (3-trifluoromethylphenyl) -2,3,5,8-tetrahydro- [ 1,2,4] triazolo [4,3-a] pyrimidin-5-yl] -phenyl} -ethyl) -2,4-dimethyl-pyridinium; 1- (2- {5-Cyano-2 - [(R) -6-methoxycarbonyl-7-methyl-3-oxo-8- (3-trifluoromethylphenyl) -2,3,5,8-tetrahydro- [ 1,2,4] triazolo [4,3-a] pyrimidin-5-yl] -phenyl} -ethyl) -3,5-dimethyl-pyridinium; 1- (2- {5-Cyano-2 - [(R) -6-methoxycarbonyl-7-methyl-3-oxo-8- (3-trifluoromethylphenyl) -2,3,5,8-tetrahydro- [ 1,2,4] triazolo [4,3-a] pyrimidin-5-yl] -phenyl} -ethyl) -2-ethylpyridinium; 1- (2- {5-Cyano-2 - [(R) -6-methoxycarbonyl-7-methyl-3-oxo-8- (3-trifluoromethylphenyl) -2,3,5,8-tetrahydro- [ 1,2,4] triazolo [4,3-a] pyrimidin-5-yl] -phenyl} -ethyl) -2- (2-hydroxy-ethyl) -pyridinium; 1-
- 来源网站:
- 中国工程科技知识中心
- 来源网址:
- http://www.ckcest.cn/home/