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(heterocycle-tetrahydropyridine) - (piperazinyl) -1-alkanone and (heterocycle dihydropyrrolidine) - (piperazinyl) -1-alkanone derivatives and their use as p75 inhibitors
专利权人:
SANOFI
发明人:
FRANÇOISE BONO,MARCO BARONI,SANDRINE DELBARY-GOSSART,VALENTINA VERCESI
申请号:
BR112012014310
公开号:
BR112012014310A2
申请日:
2010.12.13
申请国别(地区):
BR
年份:
2016
代理人:
摘要:
(heterocycle tetrahydropyridine) - (piperazinyl) -1-alkanone and (heterocycle dihydropyrrolidine) - (piperazinyl) -1-alkanone derivatives and their use as p75 inhibitors. The present invention relates to (heterocycle tetrahydropyridine) - (piperazinyl) -1-alkanone and (heterocycle dihydropyrrolidine) - (piperazinyl) -1-alkanoca derivatives of the formula (i), wherein: b, m, w, n and r 2 are as defined in claim 1, as well as the respective preparation process and its therapeutic application.derivados (heterociclo-tetra-hidropiridina)-(piperazinil)-1-alcanona e (heterociclo-di-hidropirrolidina)-(piperazinil)-1-alcanona e o respectivo uso como inibidores de p75. a presente invenção refere-se aos derivados (heterociclo-tetra-hidropiridina)-(piperazinil)-1-alcanona e (heterociclo-di-hidropirrolidina)-(piperazinil)-1-alcanoca de fórmula geral (i), na qual a,b,m,w, n e r2 são tais como definidos na reivindicação 1, assim como o respectivo processo de preparo e a respectiva aplicação em terapêutica.
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