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(Bridged piperazinyl) -1 alkanone derivatives as p75 inhibitors, their preparation process and pharmaceutical composition
专利权人:
Sanofi-Aventis
发明人:
Françoise Bono,Marco Baroni,Sandrine Delbary-Gossart
申请号:
BRPI0915126
公开号:
BRPI0915126B1
申请日:
2009.06.12
申请国别(地区):
BR
年份:
2019
代理人:
摘要:
(bridged piperazinyl) -1 alkanone derivatives as p75 inhibitors, their preparation process and pharmaceutical composition The present invention relates to ((phenyl) -3,6-dihydropyridin-1-yl) - ( bridged piperazinyl) -1-alkane and ((phenyl) -2,5-dihydro-pyrrol-1-yl) - (bridged piperazinyl) -1-alkanone of formula (i), wherein a, b, m, w, n and r 5 are as defined in claim 1, as well as the respective preparation process and its therapeutic application.derivados de (piperazinil em ponte) -1 alcanona como inibidores de p75, seu processo de preparo e composição farmacêutica a presente invenção refere-se aos derivados de ((fenil) -3,6- di-hidropiridin -1-il) - (piperazinil em ponte) -1- alcano e ((fenil) -2,5-dihidro- pirrol -1-il) - (piperazinil em ponte) -1-alcanona, de fórmula geral (i), na qual a, b, m, w, n e r5 são tais como definidos na reivindicação 1, assim como o respectivo processo de preparo e a respectiva aplicação em terapêutica.
来源网站:
中国工程科技知识中心
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