PALBOCICLIB DEUTÉRÉ

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专利权人:

CONCERT PHARMACEUTICALS INC.

发明人:

MORGAN, ADAM, J.

申请号：

EP14769343

公开号：

EP2970209A4

申请日:

2014.03.12

申请国别(地区):

EP

年份:

2016

代理人:

摘要：

The present invention refers to specifically deuterated palbociclib derivatives, wherein carbon atoms of the piperazine ring are deuterated. Like palbociclib these deuterated derivatives are cyclin-dependent kinase 4 (CDK-4) inhibitors for treating cancer. These specifically deuterated derivatives have an improved metabolic stability.

来源网站：

中国工程科技知识中心

来源网址：

http://www.ckcest.cn/home/