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Novel Selective Androgen receptor modulators
专利权人:
PFIZER INC
发明人:
PATRICK ROBERT VERHOEST,JAMES THOMAS ANDERSON,EUGENE LVOVICH PIATNITSKI CHEKLER,EDMUND L. ELLSWORTH,BRUCE KIPP ERIKCSON,ADAM MATTHEW GILBERT,ANTHONY P. RICKETTS,DAVID P. THOMPSON,RAYOMAND JAL UNWALLA
申请号:
DO2015000132
公开号:
DOP2015000132A
申请日:
2015.06.03
申请国别(地区):
DO
年份:
2015
代理人:
摘要:
The invention refers to a compound of F1, 2 or 3, wherein a is oWhere R0 is hydrogen, a linear chain tar or a branch of C1-C6, etc,Z ES –CRE––,this is it.e. Re is hydrogen, linear chain tar or C1-C6 bundle, etc;R1 is a kind of hydrogen, linear chain tar or C1-C6 bundle;R2 is independent hydrogen or tar of C1-C6 linear or branched chain, R3 and R4 are independent hydrogen, linear chain tar or C1-C6 branch, etc;R5 and R6 are hydrogen or tar independent of C1-C6 linear chain or branch;R8 is a kind of hydrogen, linear chain tar or C1-C6 beam, etc;R9 and R10 are hydrogen or tar independent of C1-C6 linear chain or branch;You need first.-Q-2-Q--it is life.Wherein, RS and RT are linear or branched chain tar independent of C1-C6, arilo, rental, heteromorphic or tar; q is 0, 1, 2, or 3; n is 0, 1, 2, 3, 4 or 5; or pharmaceutically acceptable salts of compounds containing such compounds; These compounds are used to treat various diseases, especially those affected by robot receptors or moderately infected.LA PRESENTE INVENCIÓN SE REFIERE A UN COMPUESTO DE LA FÓRMULA 1, 2 Ó 3: EN DONDE A ES N O –CR0––, DONDE R0 ES HIDRÓGENO, ALQUILO DE CADENA LINEAL O RAMIFICADA DE C1-C6, ETC., Z ES –CRE––, O, –N––, DONDE RE ES HIDRÓGENO, ALQUILO DE CADENA LINEAL O RAMIFICADA DE C1-C6, ETC.; R1 ES HIDRÓGENO, ALQUILO DE CADENA LINEAL O RAMIFICADA DE C1-C6, ETC.; R2 SON INDEPENDIENTEMENTE HIDRÓGENO O ALQUILO DE CADENA LINEAL O RAMIFICADA DE C1-C6; R3 Y R4 SON INDEPENDIENTEMENTE HIDRÓGENO, ALQUILO DE CADENA LINEAL O RAMIFICADA DE C1-C6, ETC.; R5 Y R6 SON INDEPENDIENTEMENTE HIDRÓGENO O ALQUILO DE CADENA LINEAL O RAMIFICADA DE C1-C6, ETC.; R8 ES HIDRÓGENO, ALQUILO DE CADENA LINEAL O RAMIFICADA DE C1-C6, ETC.; R9 Y R10 SON INDEPENDIENTEMENTE HIDRÓGENO O ALQUILO DE CADENA LINEAL O RAMIFICADA DE C1-C6, ETC.; Q ES ––CO––, ––(CH2)Q––, ––(CHRS)Q––, O –(CRSRT)Q––, DONDE RS Y RT SON INDEPENDIENTEMENTE ALQUILO DE CADENA LINEAL O RAMIFICADA DE C1-C6, ARILO, ALQUILARILO, HETEROARILO O ALQUILHETEROARILO; EN
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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