Jörg Kurt Wegner;Genadiy Kalayanov;Kevin Parkes;Johannes Wilhelmus J. Thuring;Wim Bert Griet Schepens;Bengt Bertil Samuelsson;Bart Rudolf Romanie Kesteleyn;Hans Kristian Wallberg
发明人:
Genadiy Kalayanov,Bart Rudolf Romanie Kesteleyn,Kevin Parkes,Bengt Bertil Samuelsson,Wim Bert Griet Schepens,Johannes Wilhelmus J. Thuring,Hans Kristian Wallberg,Jörg Kurt Wegner
申请号：
US13515187
公开号：
US08592429B2
申请日:
2010.12.10
申请国别(地区):
US
年份:
2013
代理人:
摘要：
HIV inhibitors of formula (I) wherein R1 is halo, C1-4 alkoxy, trifluoromethoxy； R2 is a group of formula (A)； R3 is a group of formula (B)； R4 is a group of formula (C)； n is 0 or 1； A is CH or N； R5 and R6 are hydrogen, C1-4 allyl, halo； R7 and R8 are C1-4 allyl or C1-4 alkoxy-C1-4 alkyl； R9 is C1-4 allyl, cyclopropyl, trifluoromethyl, C1-4 alkoxy, or dimethylamino； R10 is hydrogen, C1-4 alkyl, cyclopropyl, trifluoromethyl, C1-4 alkoxy, or dimethylamino； pharmaceutically acceptable addition salts and solvates thereof； pharmaceutical compositions containing these compounds as active ingredient and processes for preparing said compounds.
