The invention relates to compounds of formula (I): (I) R1-NH-CH(R2)-P(=O)(OH)-CH2-C(R3)(R4)-CONH-C(R5)(R6)-COOR7in which R1to R7are as defined in the claims, for the use thereof in treating and/or preventing eye inflammation, and more particularly for improving the eye healing process. Thus, the compounds of formula (I) are notably useful for preventing neovascularisation, or for preventing or treating eye inflammation linked to keratitis, scleritis, episcleritis, uveitis, a cataract, a synechia, a macular oedema, a detachment of the retina, an ocular hypertension and degeneration of the optic nerve caused by glaucoma.本發明有關於式(I)之化合物: (I) R1-NH-CH(R2)-P(=O)(OH)-CH2-C(R3)(R4)-CONH-C(R5)(R6)-COOR7其中R1至R7係如該等請求項中所界定,用於在治療及/或預防眼發炎中使用其等,且更特別地用於改善眼癒合過程。因此,式(I)之該等化合物尤其有用於預防血管增生(neovascularization),或預防或治療與角膜炎(keratitis)、鞏膜炎(scleritis)、上鞏膜炎(episcleritis)、葡萄膜炎(uveitis)、白內障、虹膜黏連(synechia)、黃斑水腫(macular oedema)、視網膜剝離、由青光眼造成的高眼壓及視神經退化相關聯的眼發炎。