OSTERKAMP FRANK,SMERLING CHRISTIANE,REINEKE ULRICH,HAASE CHRISTIAN,UNGEWISS JAN
申请号：
IN4742/DELNP/2015
公开号：
IN2015DN04742A
申请日:
2015.06.01
申请国别(地区):
IN
年份:
2015
代理人:
摘要：
The present invention is related to a compound of formula (I) wherein R1 is selected from the group consisting of hydrogen , methyl and cyclopropylmethyl AA- COOH is an amino acid selected from the group consisting of 2- amino- 2- adamantane carboxylic acid , cyclohexylglycine and 9- amino -bicyclo[3.3.1]nonane 9- carboxylic acid R2 is selected from the group consisting of (Ci- C6)alkyl , (C3- C8)cycloalkyl , (C3- C8)cycloalkylmethyl , halogen , nitro, and trifluoromethyl ALK is (C2- C5)alkylidene R3, R4 and R are each and independently selected from the group consisting of hydrogen and (Ci- C4)alkyl under the proviso that one of R3, R4 and R5 is of the formula (II) wherein ALK" is (C2- C5)alkylidene R 6is selected from the group consisting of hydrogen and (Ci- C4)alkyl and R7 is selected from the group consisting of H and an Effector moiety or a pharmacologically acceptable salt, solvate or hydrate thereof.
