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Compounds and Methods for Inhibiting CPY26 Enzymes
专利权人:
Queen's University at Kingston
发明人:
Donald Andrew Cameron,Martin Petkovich,Toni Kristian Petkovich,Victor Snieckus,Johnathan Board,Suneel Singh,Ashishkumar Jayantilal Maheta
申请号:
US16469387
公开号:
US20200093788A1
申请日:
2017.12.13
申请国别(地区):
US
年份:
2020
代理人:
摘要:
Compounds described herein are inhibitors of retinoic acid inducible P450 (CYP26) enzymes, and are useful for treating diseases that are responsive to retinoids. Certain compounds have retinoid activity, are resistant to CYP26-mediated catabolism, and are used for treating diseases that are responsive to retinoids.
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