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[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-[7-FLUORO-1-(2-METHOXY-ETHYL)-4-TRIFLUOROMETHOXY-1H-INDOL-3-YL]-METHANONE AS AN INHIBITOR OF MAST CELL TRYPTASE
专利权人:
SANOFI-AVENTIS
发明人:
CHOI-SLEDESKI, YONG MI,CHOY, NAKYEN,POLI, GREGORY BERNARD,SHAY, JR., JOHN J.,SHUM, PATRICK WAI-KWOK,SLEDESKI, ADAM W.
申请号:
MYPI 2011000395
公开号:
MY150599A
申请日:
2009.08.20
申请国别(地区):
MY
年份:
2014
代理人:
摘要:
THE PRESENT INVENTION IS DIRECTED TO AN INDOLE BENZYLAMINE COMPOUND OF FORMULA I: USEFUL AS AN INHIBITOR OF TRYPTASE. IN ADDITION, THE PRESENT INVENTION IS DIRECTED TO THE USE OF THE COMPOUND FOR TREATING A PATIENT SUFFERING FROM, OR SUBJECT TO, A PHYSIOLOGICAL CONDITION IN NEED OF AMELIORATION BY INHIBITION OF TRYPTASE, COMPRISING ADMINISTERING TO THE PATIENT OF A THERAPEUTICALLY EFFECTIVE AMOUNT OF THE COMPOUND, AND TO A PHARMACEUTICAL COMPOSITION COMPRISING A PHARMACEUTICALLY EFFECTIVE AMOUNT OF THE COMPOUND OF FORMULA I, AND A PHARMACEUTICALLY ACCEPTABLE CARRIER.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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