The present invention relates to pyrroloquinolinyl-pyrrolidine-2,5-dione compounds and methods of synthesizing these compounds. The present invention also relates to pharmaceutical compositions containing pyrroloquinolinyl-pyrrolidine-2,5-dione compounds and methods of treating cell proliferative disorders, such as cancer, by administering these compounds or pharmaceutical compositions to subjects in need thereof.本發明關於吡咯並喹啉基-吡咯啶-2,5-二酮化合物類及合成該等化合物之方法。本發明亦關於包含吡咯並喹啉基-吡咯啶-2,5-二酮化合物之醫藥組成物,及藉由投予該等化合物或醫藥組成物至需要治療之個體以治療細胞增生性疾病(諸如癌)之方法。