The present invention provides pyrroloquinolinyl-pyrrole-2,5-dione formulations and methods of treating a cell proliferative disorder, such as a cancer, by administering to a subject in need thereof a therapeutically effective amount of the formulations containing pyrroloquinolinyl-pyrrole-2,5-dione compounds.本發明提供吡咯並喹啉基-吡咯-2,5-二酮調製劑類及治療細胞增生性疾病(諸如癌症)之方法,該方法藉由投予需要治療之個體治療有效量之含有吡咯並喹啉基-吡咯-2,5-二酮化合物之調製劑。