РИНШ Кристофер (CH),ДЮПРАЗ Филиппе Виктор Леон (CH)
申请号:
RU2012106214/15
公开号:
RU2012106214A
申请日:
2010.07.23
申请国别(地区):
RU
年份:
2013
代理人:
摘要:
1. A method comprising the step of administering to a subject an amount of Punicalin, Punicalagin, Pedunculagin, Tellimagrandin, Corimagin, Granatin A, Granatine B, Termin B Terminalin), Gallagyldilactone, Compound A or a compound of Formula I: or a pharmaceutically acceptable salt, biologically active metabolite, solvate, hydrate, prodrug, enantiomer or stereoisomer thereof; wherein, independently for each case, X is or; each of R, R and R is independently hydrogen, alkyl, aralkyl, alkylcarboxy or sugar; or R represents hydrogen, alkyl, aralkyl, alkyl carboxy, or sugar, R represents hydrogen or, and R represents; or R is hydrogen, alkyl, aralkyl, alkyl carboxy or sugar, and R and R together are 2. The method according to claim 1, characterized in that X represents 3. The method according to claim 1, characterized in that X represents 4. The method according to claim 1, wherein R is hydrogen. The method according to claim 1, wherein R is a sugar selected from the group consisting of allose ("All"), altrose ("Alt"), arabinose ("Ara"), erythrose, erythrulose, fructose ("Fru" ), fucosamine ("FucN"), fucose ("Fuc"), galactosamine ("GalN"), galactose ("Gal"), galloyl-β-glucose, glucosamine ("GlcN"), glucosaminite ("GlcN-ol" ), glucose (“Glc”), glyceraldehyde, 2,3-dihydroxypropanal, glycerol (“Gro”), propane-1,2,3-triol, glyceron (“1,3-dihydroxyacetone”), 1,3-dihydroxypropanone , guloses ("Gul"), idoses ("Ido"), lyxoses ("Lyx"), mannosamine ("ManN"), mannose ("Man"), psychosis ("Psi"), hin wagons ( «Qui»), hinovozamina, ramnita ( «Rha-ol»), ramnozamina ( «RhaN»), rhamnose ( «Rha»), ribose ( «Rib»), ri1. Способ, включающий этап введения субъекту количества Пуникалина (Punicalin), Пуникалагина (Punicalagin), Педункулагина (Pedunculagin), Теллимаграндина (Tellimagrandin), Корилагина (Corilagin), Гранатина A (Granatine А), Гранатина Б (Granatine В), Терминалина (Terminalin), Галлагилдилактона (Gallagyldilactone), Соединения А или соединения Формулы I:или его фармацевтически п