FORSCHUNGSVERBUND BERLIN E.V.;LUDWIG-MAXIMILIANS-UNIVERSITAT MUNCHEN
发明人:
CHRISTIAN, HACKENBERGER,KASPER, MARC ANDRE,GLANZ, MARIA,SAUER, TOM,SCHUMACHER, DOMINIK,HELMA-SMETS, JONAS,LEONHARDT, HEINRICH,STENGL, ANDREAS
申请号:
CA3032251
公开号:
CA3032251A1
申请日:
2017.09.01
申请国别(地区):
CA
年份:
2018
代理人:
摘要:
Disclosed are novel conjugates and processes for the preparation thereof. A process for the preparation of alkene- or alkyne-phosphonamidates comprises the steps of (I) reacting a compound of formula (III), with an azide of formula (IV), to prepare a compound of formula (V), reacting a compound of formula (V) with a thiol-containing molecule of formula (VI), resulting in a compound of formula (VII).