LUDWIG-MAXIMILIANS-UNIVERSITÄT MÜNCHEN;FORSCHUNGSVERBUND BERLIN E.V.
发明人:
Christian Hackenberger,Marc André Kasper,Maria Glanz,Tom Sauer,Dominik Schumacher,Jonas Helma-Smets,Heinrich Leonhardt,Andreas Stengl
申请号：
US16328199
公开号：
US20190330264A1
申请日:
2017.09.01
申请国别(地区):
US
年份:
2019
代理人:
摘要：
Disclosed are novel conjugates and processes for the preparation thereof. A process for the preparation of alkene- or alkyne-phosphonamidates comprises the steps of (I) reacting a compound of formula (III), with an azide of formula (IV), to prepare a compound of formula (V), reacting a compound of formula (V) with a thiol-containing molecule of formula (VI), resulting in a compound of formula (VII).
