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sphingosine kinase inhibitors
专利权人:
MERCK PATENT GMBH
发明人:
DIRK WIENKE,FRANK STIEBER
申请号:
BR112012014884
公开号:
BR112012014884A2
申请日:
2010.11.18
申请国别(地区):
BR
年份:
2016
代理人:
摘要:
Sphingosine kinase inhibitors The invention relates to compounds of formula (I), wherein R1, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11, R12, R13, R14, R15, R16 , r17, m1, m2, m3, m4, y1, y2, v, w, n, mes have the meanings specified herein, and their physiologically compatible salts, derivatives, prodrugs, solvates, tautomers and stereoisomers thereof, including their mixtures in all proportions for use in the treatment of diseases that are influenced by inhibiting efingosine kinase 1.inibidores de esfingosina quinase a invenção refere-se a compostos de fórmula (i), em que r1, r2, r3, r4, r5, r6, r7, r8, r9, r10, r11, r12, r13, r14, r15, r16, r17, m1, m2, m3, m4, y1, y2, v, w, n, m e s têm os significados aqui especificados, e aos seus sais fisiologicamente compatíveis, derivados, prodrogas, solvatos, tautômeros e estereisômeros do mesmo, incluindo as suas misturas em todas as proporções, por usar no tratamento de doenças que são influenciadas pela quinase a efingosina de inibição 1.
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