PHILIP DR. LIENAU,ALEXANDER PROF. DR. HILLISCH,CHRISTOPH DR. GERDES,MICHAEL DR. GERISCH,TOM DR. KINZEL,KAREN DR. ENGEL,ANJA DR. BUCHMLLER,SUSANNE DR. RHRIG,MARTINA VICTORIA DR. SCHMIDT,JULIA STRABURGE
申请号：
ARP140102148
公开号：
AR096516A1
申请日:
2014.05.30
申请国别(地区):
AR
年份:
2016
代理人:
摘要：
Claim 1: Compound of the formula (1) in which r u00b9 represents a group of formulas (2) which is the point of attachment to the carbonyl Group； X represents an oxygen Atom or a Sulfur Atom, Ch r u2076, where r u2076 represents R u00b2 alqui represents Hydrogen, hydroxyl； The c u2081 u208b u2086, cycloalkyl or c u2083 u208b u2086 phenylWhere can be substituted with alkyl and cycloalkyl a Substituent selected from the group consisting of Hydroxy, methoxy, cyano, hidroxicarbonilo, aminocarbonilo, metilsulfonilo Difluoromethoxy and trifluoromethoxy, or alkyl and cycloalkyl substituted with 1 to 3 can be replaced Total Fluorine； r u00b3 represents Hydrogen or alkyl c u2081 u208b u2084,Or R u00b2 and r u00b3 along with the carbon Atom to which they are United to form a Ring ciclopropilo, ciclobutilo Cyclopentyl Ring or ring, the ring and the ciclobutilo Cyclopentyl Ring may be substituted with a hydroxyl Substituent； r u2074 represents Hydrogen or alqui The c u2081 u208b u2086, where Rent can be substituted with a hydroxyl Substituent is alkyl； r u2075 c u2081 u208b u2084,Or r u2074 and r u2075 along with the carbon Atom to which they are United to form a Ring ciclopropilo, ciclobutilo Cyclopentyl Ring or ring, the ring and the ciclobutilo Cyclopentyl Ring may be substituted with a hydroxyl Substituent； r u2077 represents Hydrogen or alkyl Or c u2081 u208b u2086, where Rent can be substituted with a hydroxyl Substituent or cyano,Or where Rent can be substituted with 1 to 3 r u2078 represents Fluorine substituents； Hydrogen； r u2079 represents Hydrogen or alkyl c u2081 u208b u2086, where Rent can be substituted with a hydroxyl Substituent or cyano, or where Rent can be substituted with 1 to 3 r u00b9 Fluorine substituents. u2070 represents Hydrogen, alkyl r u00b9 u00b9 represents c u2081 u208b u2084,Where Rent can be substituted with a hydroxyl Substituent； r u00b9 u00b2 represents Hydrogen or alkyl c u2081 u208b u2084, or r u00b9 u00b9 and r u00b9 u00b2 along with the c
