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MACROCYCLIC BROAD SPECTRUM ANTIBIOTICS
专利权人:
RQX PHARMACEUTICALS, INC.;GENENTECH, INC.
发明人:
SMITH, Peter,ROBERTS, Tucker,HIGUCHI, Robert,PARASELLI, Prasuna,KOEHLER, Michael,SCHWARZ, Jacob,CRAWFORD, James,LY, Cuong Q.,HANAN, Emily,HU, Huiyong,CHEN, Yongsheng,YU, Zhiyong,Paul Colin Michael Win
申请号:
SG11201907448R
公开号:
SG11201907448RA
申请日:
2018.02.22
申请国别(地区):
SG
年份:
2019
代理人:
摘要:
INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (43) International Publication Date 23 August 2018 (23.08.2018) WIP0 I PCT 0111111010 0111 °nolo Holum° mumionio oimIE (10) International Publication Number WO 2018/149419 Al (51) International Patent Classification: CO7D 245/04 (2006.01) A61P 31/04 (2006.01) A61K 31/395 (2006.01) (21) International Application Number: PCT/CN2018/076957 (22) International Filing Date: 22 February 2018 (22.02.2018) (25) Filing Language: English (26) Publication Language: English (30) Priority Data: PCT/CN2017/073575 15 February 2017 (15.02.2017) CN PCT/CN2017/085075 19 May 2017 (19.05.2017) CN (71) Applicants: RQX PHARMACEUTICALS, INC. [US/US]; 11099 N. Torrey Pines Road, Suite 290, La Jolla, CA 92037 (US). GENENTECH, INC. [US/US]; 1 DNA Way, South San Francisco, CA 94080 (US). (72) Inventors: SMITH, Peter, Andrew; 260 King Street Unit 909, San Francisco, CA 94107 (US). ROBERTS, Tuck- er, Curran; 536 Maple Street, Apt. 301, San Diego, CA 92103 (US). HIGUCHI, Robert, I.; 434 Marview Dri- ve, Solana Beach, CA 92075 (US). PARASELLI, Pra- suna; 6323 Oleander Way, San Diego, CA 92130 (US). KOEHLER, Michael, F., T.; 516 Georgia Avenue, Pa- lo Alto, CA 94306 (US). SCHWARZ, Jacob, Bradley; 7211 Balmoral Way, San Ramon, CA 94582 (US). CRAW- FORD, James, John; 1501 Church St #102, San Fran- cisco, CA 94131 (US). LY, Cuong Q.; 801 Maple Av- enue, Burlingame, CA 94010 (US). HANAN, Emily, J.; 1904 Woodside Road, Redwood City, CA 94061 (US). HU, Huiyong; 34121 Susa Terrace, Fremont, CA 94555 (US). CHEN, Yongsheng; 288 Fute Zhong Road, Waigao- qiao Free Trade Zone, Shanghai 200131 (CN). YU, Zhiy- ong; 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131 (CN). (74) Agent: AFD CHINA INTELLECTUAL PROPERTY LAW OFFICE; Suite B 1601A, 8 Xue Qing Road, Haidi- an, Beijing 100192 (CN). (81) Designated States (unless otherwise indicated, for every kind o
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