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STAT3/5 ACTIVATION INHIBITOR
专利权人:
OTSUKA PHARMACEUTICAL CO.; LTD.
发明人:
SEKIGUCHI, KAZUO,SUGIYAMA, KAZUHISA,AKAMATSU, SEIJI,KIYONO, KUNIHIKO,YANAGIHARA, YASUO,WATANABE, TAKASHI,HAYASHI, KAZUHIKO,TANAKA, HIDEO,SUMIDA, TAKUMI,SUZUKI, TAKASHI,OHBUCHI, YUTAKA,OKUNO, MITSUHIRO
申请号:
MYPI 20091324
公开号:
MY150229A
申请日:
2007.10.02
申请国别(地区):
MY
年份:
2013
代理人:
摘要:
AN OBJECT OF THE PRESENT INVENTION IS TO PROVIDE A STAT3/5 ACTIVATION INHIBITOR. THE PRESENT INVENTION PROVIDES A STAT3/5 ACTIVATION INHIBITOR CONTAINING AN AROMATIC COMPOUND REPRESENTED BY THE GENERAL FORMULA OR A SALT THEREOF AS AN ACTIVE INGREDIENT: WHEREIN X₁ REPRESENTS A NITROGEN ATOM OR A GROUP -CH=, R₁ REPRESENTS A GROUP -Z-R⁶, IN WHICH Z REPRESENTS A GROUP -CO-, A GROUP -CH(OH)- OR THE LIKE, R6 REPRESENTS A 5-TO 15-MEMBERED MONOCYCLIC, DICYCLIC OR TRICYCLIC SATURATED OR UNSATURATED HETEROCYCLIC GROUP HAVING 1 TO 4 NITROGEN ATOMS, OXYGEN ATOMS OR SULFUR ATOMS, R² REPRESENTS A HYDROGEN ATOM OR A HALOGEN ATOM, Y REPRESENTS A GROUP -C-, A GROUP -CO-, A GROUP -CH(OH)- OR A LOWER ALKYLENE GROUP, AND A REPRESENTS A GROUP WHEREIN R³ REPRESENTS A HYDROGEN ATOM, A LOWER ALKOXY GROUP OR THE LIKE, P REPRESENTS 1 OR 2, R⁴ REPRESENTS AN IMIDAZOLYL LOWER ALKYL GROUP OR THE LIKE.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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