NIELSEN, MOGENS,LILJEFORS, TOMMY,NILSSON, JAKOB,STERNER, OLOV
申请号：
CA2720461
公开号：
CA2720461C
申请日:
2009.04.02
申请国别(地区):
CA
年份:
2016
代理人:
摘要：
The present invention relates to novel GABA A /BzR ligands of the generalformulas (I), (II) and (III) wherein R1 isselected from the group consisting of hydrogen, halogen, haloalkyl having 1-2carbon atoms, alkoxy having 1 to 3 carbon atoms inthe alkyl chain, alkyl having 1 to 3 carbon atoms, and nitro, and R2 isselected from the group consisting of hydrogen, halogen andalkyl having 1 to 2 carbon atoms, as well as the use of these compounds fortreating anxiolytic, anticonvulsant, sedative- hypnoticand myorelaxant conditions as well as anxiogenic, somnolytic and convulsantconditions in mammals including pharmaceuticalcompositions comprising the same
