The invention relates to a composition for the treatment of the organelles of genetically healthy cells of human beings, particularly for preventive treatment of the cells supporting control system, comprising at least one active agent having strong competitively binding hormone antagonist properties combined with at least a first and/or a second carrier medium supporting the transport of molecules of said active agent through the cell-wall into the cytosol and organelles of cells. In preferred forms of applications, groups of at least a first and a second inventive composition are provided that comprise different carrier media and that are applicable in different parts of the body for forwarding the active agent via different pathways to a determined application zone.