BAYER CROPSCIENCE AKTIENGESELLSCHAFT;BAYER AKTIENGESELLSCHAFT;BAYER ANIMAL HEALTH GMBH;BAYER PHARMA AKTIENGESELLSCHAFT
发明人:
JANSSEN, ISA JANA IRINA,DR. HEISLER, IRING,DR. ALIG, BERND,DR. HBSCH, WALTER,GRGENS, ULRICH,DR. HALLENBACH, WERNER,DR. SCHWARZ, HANS,GEORG - PROF. DR. ILG, THOMAS,DR. BRNGEN, KIRSTEN,DR. BHM, CLAUDIA
申请号:
ARP180101808
公开号:
AR112216A1
申请日:
2018.06.29
申请国别(地区):
AR
年份:
2019
代理人:
摘要:
These compounds are intermediate compounds that can be used to prepare these compounds, their preparation procedures, including the compounds and combinations of these compounds, as well as pharmaceutical compounds for treatment using these compounds, Control and / or prevent disease, especially worm infection, as a single vector or in combination with other active ingredients. 1. Claim 1: compound (1) of general formula,A is the compound of formula (2) or (3);o is 0, 1, 2, 3 or 4; R is selected from the group consisting of hydrogen, halogen, cyano, nitro, -OH, C--alkyl,a. Halogen-c83216c83318324, including 1 to 5 halogen atoms, alcox-c83218c83124;halogenoalkoxy-C₁₋₄ having 1 to 5 halogen atoms, cycloalkyl-C₃₋₆,-NH832222,-NH (C--alkyl),-N (alkyl-C₁₋₄) ₂,-S-rental - c8321c83318324;-S (o) - rental - c8332124;-SO₂-alkyl-C₁₋₄,-S-halogenalkyl-C₁₋₄,-S (O) -halogenalkyl-C₁₋₄ and -SO₂-halogenalkyl-C₁₋₄ having 1 to 5 halogen atoms; X, Y are independently selected from the group consisting of CR⁷R⁸,O. S, and n-r8313,The feature is that at least one of X and Y is cr8311; r831222,If you are already registered, please log in first.-C (o) - No. 8313-S (o) - No. 8313-SO₂-NR⁹- and -SO₂-O-;T selected from the formula group (4);R¹ is selected from the group consisting of hydrogen, cyano, -CHO, -OH, alkyl-C₁₋₄,a. Halogen-c83216c83318324, including 1 to 5 halogen atoms, alcox-c83218c83124;halogenoalkoxy-C₁₋₄ having 1 to 5 halogen atoms, cycloalkyl-C₃₋₆,a. Halogenated CYCLOPROPYLENE glycol-c83231;alkynyl-C₃₋₄,alkoxy-C₁₋₄-alkyl-C₁₋₄,cycloalkyl-C₃₋₆-alkyl-C₁₋₃,cyano-C₁₋₄-alkyl, -NH-alkyl-C₁₋₄,-N (alkyl-C₁₋₄) ₂,Nhc23222-let-c832131;C--alkyl-NH-C₁₋₄-alkyl,1.A.1.a.1.1.b.1.1.1.1.a.1.b1. Asphalt-c83218c83331-83224c (o) -,a. Halogen-c83217c83318324c (o) - consists of one to five halogen atoms, alcox-c83321c83318324c (o) -;Datum-c (o)alcoxi-C -alquilo-C -C (O) --SO₂-alkyl-C₁₋₄,and -SO₂-halogenoalkyl-C₁₋₄ having 1 to 5 halogen atoms; phenyl-C₁₋₄-alkyl, optionally substituted by 1, 2, 3, 4 or 5 su