Андрей Александрович,Александр Васильевич,Володимир Михайлович,Олег Дмитриевич,Николай Филиппович
申请号：
EA201101327
公开号：
EA201101327A1
申请日:
2010.04.30
申请国别(地区):
EA
年份:
2012
代理人:
摘要：
the invention relates to a new \u0437\u0430\u043c\u0435\u0449\u0435\u043d\u043d\u044b\u043c 8 - sulfonyl - 2,3,4,5-tetrachlorophenol of 1h - gamma \u043a\u0430\u0440\u0431\u043e\u043b\u0438\u043d\u0430\u043c general formula 1 and their \u0444\u0430\u0440\u043c\u0430\u0446\u0435\u0432\u0442\u0438\u0447\u0435\u0441\u043a\u0438 acceptable salts - \u043b\u0438\u0433\u0430\u043d\u0434\u0430\u043c,at the same time with biological activity against alpha \u0430\u0434\u0440\u0435\u043d\u043e\u0446\u0435\u043f\u0442\u043e\u0440\u043e\u0432, \u0434\u043e\u043f\u0430\u043c\u0438\u043d\u043e\u0432\u044b\u0445 receptors antagonist, \u0438\u043c\u0438\u0434\u0430\u0437\u043e\u043b\u0438\u043d\u043e\u0432\u044b\u0445 \u0440\u0435\u0446\u0435\u043f\u0442\u043e\u0440\u043e the sigma receptor\u043d\u043e\u0440\u0435\u043f\u0438\u043d\u0435\u0444\u0440\u0438\u043d\u0435\u0432\u044b\u0445 \u0441\u0435\u0440\u043e\u0442\u043e\u043d\u0438\u043d\u043e\u0432\u044b\u0445 receptors, receptors for active component, pharmaceutical compositions containing, as an active component, a new l \u0438\u0433\u0430\u043d\u0434\u044b to new medicines.used for the treatment of diseases and conditions of the central nervous system. in the general formula 1.r1 represents a deputy chosen from hydrogen, optionally \u0437\u0430\u043c\u0435\u0449\u0435\u043d\u043d\u043e\u0433\u043e c1 - c3 \u0430\u043b\u043a\u0438\u043b\u0430 or c1 - c4 \u0430\u043b\u043a\u0438\u043b\u043e\u043a\u0441\u0438\u043a\u0430\u0440\u0431\u043e\u043d\u0438\u043b\u0430 r2 represents the \u0446\u0438\u043a\u043b\u0438 delivery systemincluding hydrogen atom, optionally \u0437\u0430\u043c\u0435\u0449\u0435\u043d\u043d\u044b\u0439 c1 - c3 \u0430\u043b\u043a\u0438\u043b,not necessarily \u0437\u0430\u043c\u0435\u0449\u0435\u043d\u043d\u044b\u0439 c2 - c3 \u0430\u043b\u043a\u0435\u043d\u0438\u043b or \u0437\u0430\u043c\u0435\u0449\u0435\u043d\u043d\u044b\u0439 sulfonyl r3 represents optionally \u0437\u0430\u043c\u0435\u0449\u0435\u043d\u043d\u0
