GENENTECH, INC.;CONSTELLATION PHARMACEUTICALS, INC.
发明人:
Brian K. Albrecht,Steven F. Bellon,Daniel J. Burdick,Alexandre Cote,Terry Crawford,Les A. Dakin,Vickie Hsiao-Wei Tsui,Michael Charles Hewitt,Yves LeBlanc,Steven R. Magnuson,Christopher G. Nasveschuk,A
申请号:
US15592017
公开号:
US10150767B2
申请日:
2017.05.10
申请国别(地区):
US
年份:
2018
代理人:
摘要:
The present invention relates to compounds of formula (I):and to salts thereof, wherein R1, R2, and Q have any of the values defined in the specification, and compositions and uses thereof. The compounds are useful as inhibitors of bromodomains. Also included are pharmaceutical compositions comprising a compound of formula (I) or a pharmaceutically acceptable salt thereof, and methods of using such compounds and salts in the treatment of various bromodomain-mediated disorders.