TRIAMIDES D'ACIDE N-PHENYL-PHOSPHORIQUE, PROCEDES POUR LES PRODUIRE ET LEUR UTILISATION COMME AGENTS POUR REGULER OU INHIBER L'HYDROLYSE ENZYMATIQUE DE L'UREE
The invention relates to N-phenylphosphonic acid triamides of general formula(I), to a method for the production thereof and to their use as agents forregulating or inhibiting enzymatic urea hydrolysis. In formula (I), Xrepresents oxygen or sulfur； R1, R2, R3, R4, R5, independent of one another,represent hydrogen C1-C8 alkyl/heteroalkyl, C2-C8 alkenyl/heteroalkenyl, C2-C8-alkynyl/heteroalkynyl, C3-C8 cycloalkyl/heterocycloalkyl, C3-C8cycloalkenyl/heterocycloalkenyl, C6-C10 aryl/C5-C10 heteroaryl, aralkyl,heteroarylalkyl, alkaryl, alkheteroaryl, alkoxy, aryloxy, hetaryloxy,alkylthio, arylthio, hetarylthio, acyl, aroyl, hetaroyl, acyloxy, aroyloxy,hetaroyloxy, alkoxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl,alkylsulfonyl, fluorine, chlorine, bromine, iodine, cyano, nitro, sulfo,carbonyl, carboxy, carbamoyl, sulfamoyl, with the provision that: at least oneradical R is not hydrogen； in the event R1, R2, R4, R5 represent H, R3 is notnitro or cyano, and； in the event R1 represents Cl or R1 and R3 represent Cl,at least one of the remaining radicals is not hydrogen.
