JONCKERS, TIM HUGO MARIA,DIERYNCK, INGE,LAST, STEFAAN JULIEN,DE KOCK, HERMAN
申请号:
CA2651659
公开号:
CA2651659C
申请日:
2007.05.30
申请国别(地区):
CA
年份:
2014
代理人:
摘要:
The present invention concerns lysine related derivatives of Formula (I)(see formula I)their use as protease inhibitors, in particular as HIV aspartyl proteaseinhibitors, processes fortheir preparation as well as pharmaceutical compositions and diagnostic kitscomprisingthem. The present invention also concerns combinations of the present lysinerelatedderivatives with another anti-retroviral agent. It further relates to theiruse in assays asreference compounds or as reagents.