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DERIVADOS DE AZAQUINOLIN-CARBOXAMIDA
专利权人:
MERCK PATENT GMBH
发明人:
HUCK, BAYARD,LAN, RUOXI,POTNICK, JUSTIN,DESELM, LIZBETH CELESTE,CRONIN, JR., MARK,NEAGU, CONSTANTIN,CHEN, XIAOLING,BOIVIN, ROCH,JOHNSON, THERESA L.,GOUTOPOULOS, ANDREAS
申请号:
PE0006932015
公开号:
PE17822015A1
申请日:
2013.11.27
申请国别(地区):
PE
年份:
2015
代理人:
摘要:
Refers to azaquinazolin - carboxamide Derivatives of formula (i) wherein R1, R2, R3, W1, W2, W3, W4 and M are as defined in the description. Preferred compounds are: 4 - (3 - trifluoromethyl - Benzylamino) - benzo [d] [1,2,3] triazin - 8 - carboxamide 4 - ((4 - diclorobencil) amino) benzo [d] [1,2,3] triazin - 8 - carboxamide among others. It also relates to a Pharmaceutical composition.These compounds are inhibitors of p70S6K is useful for the treatment of hiperproliferativos Disorders such as cancer, gliomaSE REFIERE A DERIVADOS DE AZAQUINAZOLIN-CARBOXAMIDA DE FORMULA (I) DONDE R1, R2, R3, W1, W2, W3, W4 Y m SON TAL COMO SE DEFINEN EN LA DESCRIPCION. SON COMPUESTOS PREFERIDOS: 4-(3-TRIFLUOROMETIL-BENCILAMINO)-BENZO[d][1,2,3]TRIAZIN-8-CARBOXAMIDA 4-((3,4-DICLOROBENCIL)AMINO) BENZO[d][1,2,3]TRIAZIN-8-CARBOXAMIDA ENTRE OTROS. TAMBIEN SE REFIERE A UNA COMPOSICION FARMACEUTICA. DICHOS COMPUESTOS SON INHIBIDORES DE P70S6K SIENDO UTILES PARA EL TRATAMIENTO DE TRASTORNOS HIPERPROLIFERATIVOS COMO CANCER, GLIOMA
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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