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INDAZOLYL THIADIAZOLAMINES AND RELATED COMPOUNDS FOR INHIBITION OF RHO-ASSOCIATED PROTEIN KINASE AND THE TREATMENT OF DISEASE
专利权人:
发明人:
Thomas Daniel Aicher,Fernando Padilla,Peter L. Toogood,Shoujun Chen
申请号:
US15551132
公开号:
US20180093978A1
申请日:
2016.02.26
申请国别(地区):
US
年份:
2018
代理人:
摘要:
The invention provides indazolyl thiadiazolamines and related compounds, pharmaceutical compositions, methods of inhibiting Rho-associated protein kinase, and methods of treating inflammatory disorders, immune disorders, fibrotic disorders, and other medical disorders using such compounds. An exemplary indazolyl thiadiazolamine compound is an N-(5-[5-[(1H4ndazol-5-yl)amino]-1,3,4-thiadiazol-2-yl]pyridin-3-yl)acetamide compound.
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中国工程科技知识中心
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http://www.ckcest.cn/home/

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