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Isothiazolopyrimidinones, pyrazolopyrimidinones, and pyrrolopyrimidinones as ubiquitin-specific protease 7 inhibitors
专利权人:
Inc.;Forma Therapeutics
发明人:
Stephanos Ioannidis,Adam Charles Talbot,Bruce Follows,Alexandre Joseph Buckmelter,Minghua Wang,Ann-Marie Campbell
申请号:
US15015566
公开号:
US09938300B2
申请日:
2016.02.04
申请国别(地区):
US
年份:
2018
代理人:
摘要:
The disclosure relates to inhibitors of USP7 inhibitors useful in the treatment of cancers, neurodegenerative diseases, immunological disorders, inflammatory disorders, cardiovascular diseases, ischemic diseases, viral infections and diseases, and bacterial infections and diseases, having the Formula:where R1, R2, R3, R4, R5, R5′, X1, X2, X3, n, and m are described herein.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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